Affinity DataKi: 3.30E+3nMAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki=IC50/(1+[L]/Kd] where [L] is the concentration of labeled ligand a...More data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki=IC50/(1+[L]/Kd] where [L] is the concentration of labeled ligand a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [3H]R5020 binding to cytosolic progesterone receptor (PRc) of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of [3H]R5020 binding to cytosolic progesterone receptor (PRc) of rat uterusMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of [3H]R5020 binding to cytosolic progesterone receptor (PRc) of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 7.43nMAssay Description:Inhibitory progestational activity on oral administration in uterine C3 modelMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of [3H]R5020 binding to cytosolic progesterone receptor (PRc) of rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 67.3nMAssay Description:Inhibitory progestational activity on oral administration in uterine C3 modelMore data for this Ligand-Target Pair
Affinity DataIC50: 92.5nMAssay Description:Effective concnetration against Androgen receptor in mouse fibroblast L929 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 942nMAssay Description:Effective concentration of progesterone receptor agonist induction of alkaline phosphatase activity in human T47D breast carcinoma cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibitory progestational activity on oral administration in uterine C3 modelMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Binding affinity to progesterone receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Binding affinity to progesterone receptorMore data for this Ligand-Target Pair
